Rimonabant-d10

SI-7687

Rimonabant-d₁₀, >98% (HPLC)

CAS No. : [929221-88-5]

Synonyms : SR-141716-d₁₀

IUPAC Name : 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl-d₁₀)-1H-pyrazole-3-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Rimonabant‑d₁₀ is a deuterium labelled version of Rimonabant, enabling enhanced analytical detection and pharmacokinetic profiling. Rimonabant itself is a highly potent, brain‑penetrant CB1 receptor antagonist (K_i = 1.8 nM) with secondary inhibitory activity against the mycobacterial membrane protein MMPL3.

References : Russak E. M. et al.: Ann Pharmacother. 53(2), 211-216, 2019; Leite C. E. et al.: Pharmacol. Rep., 61, 217-224, 2009; Seely K. A. et al.: Neuropharmacology, 63(5), 905-15, 2012; Zhang B. et al.: Cell, 176(3), 636-648, 2019; Erdozain A. M. et al.: Biochem Pharmacol, 83(2), 260-268, 2012.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.