Rociletinib

SI-2483

Rociletinib, >98% (HPLC)

CAS No. : [1374640-70-6]

MDL No. : MFCD26793864

Synonyms : CO-1686; AVL-301; CNX-419

IUPAC Name : N-(3-((2-((4-(4-Acetylpiperazin-1-yl)-2-methoxyphenyl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	85.00		Back Order	Estimated to ship on 04 October 2026
50MG	135.00		Back Order	Estimated to ship on 04 October 2026
100MG	235.00		Back Order	Estimated to ship on 04 October 2026
250MG	455.00		Back Order	Estimated to ship on 04 October 2026
500MG	855.00		Back Order	Estimated to ship on 04 October 2026

Applications : A potent, highly selective, irreversible inhibitor of mutant EGFR with Ki of 21.5 nM for EGFR ^L858R/T790M.

References : Walter A. O. et al.: Cancer Discov., 3(12), 1404-1415, 2013; Tjin Tham Sjin R. et al.: Mol Cancer Ther.,13(6), 1468-1479, 2014; Sequist L. V. et al.: N Eng. J. Med., 372(18), 1700-1709, 2015.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.