(S)-GSK-852

SI-6758

(S)-GSK-852, >98% (HPLC)

CAS No. : [2305919-51-9]

IUPAC Name : (S)-N5-((1R,3S,5S,6r)-3-Hydroxybicyclo[3.1.0]hexan-6-yl)-N7,3-dimethyl-3-phenyl-2,3-dihydrobenzofuran-5,7-dicarboxamide

Price And Availability
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5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
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Applications : (S)-GSK-852 represents the (S)‑diastereomer of GSK-852, a BET inhibitor that preferentially targets the second bromodomain (BD2) with a pIC₅₀ of 7.9. The diastereomer supports studies examining the impact of chirality on BD2‑selective BET engagement.

References : Lucas S. C. C. et al.: J. Med. Chem., 64(15), 10711-10741, 2021.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.