Serabelisib

SI-5337

Serabelisib, >98% (HPLC)

CAS No. : [1268454-23-4]

MDL No. : MFCD15146372

Synonyms : MLN1117; INK1117; TAK-117

IUPAC Name : (6-(2-Aminobenzo[d]oxazol-5-yl)imidazo[1,2-a]pyridin-3-yl)(morpholino)methanone

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
1G	Request A Quote		Back Order	Estimated to ship on 04 October 2026
5G	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10G	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Serabelisib is a potent and selective oral PI3Kα isoform inhibitor (IC50 of 21 nmol/L against PI3Kα) that has demonstrated > 100-fold selectivity relative to other class I PI3K family members (PI3Kβ/γ/δ) and mTOR, and a high degree of selectivity against many other kinase. Potential antineoplastic activity.

References : Juric D. Clin Cancer Res., 23(17), 5015-5023, 2017; Yea S. S. et al.: PLoS One, 9(6), e99486, 2014; Katti Jessen et al.: AACR; Mol Cancer Ther., 10(11 Suppl):Abstract nr A171, 2011.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.