Sitagliptin

SI-4508

Sitagliptin, >98% (HPLC)

CAS No. : [486460-32-6]

MDL No. : MFCD09838015

Synonyms : MK-0431; MK0431

IUPAC Name : (R)-3-Amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-4-(2,4,5-trifluorophenyl)butan-1-one

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
1G	15.00		In Stock	Estimated to ship on 20 September 2026
5G	25.00		In Stock	Estimated to ship on 20 September 2026
10G	35.00		In Stock	Estimated to ship on 20 September 2026
25G	65.00		In Stock	Estimated to ship on 20 September 2026
100G	215.00		In Stock	Estimated to ship on 20 September 2026

Applications : Sitagliptin is an oral and highly selective DPP-4 inhibitor with an IC₅₀ of 18 nM. It is used for the treatment of type 2 diabetes.

References : Karasik A. et al.: Curr Med Res Opin., 24(2), 489-496, 2008; Kim S. J. et al.: Diabetes 58(3), 641-651, 2009; Sangle G. V. et al.: Endocrinology 153(2), 564-573,2012.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.