SR-48692

SI-7650

SR-48692, >98% (HPLC)

CAS No. : [146362-70-1]

Synonyms : Meclinertant; SR-48692

IUPAC Name : (1r,3r,5r,7r)-2-(1-(6-Chloroquinolin-4-yl)-5-(2,6-dimethoxyphenyl)-1H-pyrazole-3-carboxamido)adamantane-2-carboxylic acid

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : SR-48692 is an orally active, nonpeptidic NTSR1 antagonist with sub‑nanomolar potency (IC₅₀= 0.99 nM) and no detectable agonist effects. Its pharmacological profile supports its use in studies of neurotensin‑regulated neurotransmission and behavior.

References : Dubuc I. et al.: Br. J. Pharmacol., 112(2), 352-4, 1994; Steinberg R. et al.: Neuroscience, 59(4), 921-9, 1994; Brouard A. et al.: Eur. J. Pharmacol., 253(3), 289-91, 1994; Gully D. et al.: Proc. Natl. Acad. Sci. U S A., 90(1), 65-9, 1993.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.