SRX-246

SI-7483

SRX-246, >98% (HPLC)

CAS No. : [512784-93-9]

IUPAC Name : (R)-4-([1,4'-Bipiperidin]-1'-yl)-4-oxo-2-((3S,4R)-2-oxo-3-((S)-2-oxo-4-phenyloxazolidin-3-yl)-4-((E)-styryl)azetidin-1-yl)-N-((S)-1-phenylethyl)butanamide

Price And Availability
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5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
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Applications : SRX-246 potently and selectively inhibits the human V1a receptor (K_i = 0.3 nM) and shows no interaction with V1b or V2 receptors. It also exhibits minimal off‑target binding across 64 receptor classes. With strong BBB penetration and high selectivity, SRX-246 is a valuable tool for studying V1a‑dependent pathways in stress‑related disease models.

References : Guillon C. D. et al.: Bioorg. Med. Chem., 15(5), 2054-80, 2007; Fabio K. M. et al.: J. Pharm. Sci., 102(6), 2033-2043, 2013.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.