Tanzisertib

SI-6883

Tanzisertib, >98% (HPLC)

CAS No. : [899805-25-5]

Synonyms : CC-930

IUPAC Name : (1S,4r)-4-((9-((S)-Tetrahydrofuran-3-yl)-8-((2,4,6-trifluorophenyl)amino)-9H-purin-2-yl)amino)cyclohexan-1-ol

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Tanzisertib potently inhibits all three JNK isoforms, with IC₅₀ values of 61 nM (JNK1), 7 nM (JNK2), and 6 nM (JNK3). It is widely used to probe JNK‑mediated pathways in inflammation, fibrosis, and stress‑response signaling.

References : Lay T. Gan et al.: J. Hepatol., 61(6), 1376-84, 2014; Nicole Reich et al.: Ann Rheum Dis., 71(5), 737-45, 2012.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.