Tersolisib

SI-7591

Tersolisib, >98% (HPLC)

CAS No. : [2883540-92-7]

Synonyms : LY-4064809; STX-478-101; STX-478

IUPAC Name : (R)-1-(2-Aminopyrimidin-5-yl)-3-(1-(5,7-difluoro-3-methylbenzofuran-2-yl)-2,2,2-trifluoroethyl)urea

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Tersolisib selectively inhibits mutant PI3Kα through an allosteric mechanism and shows excellent oral exposure and CNS penetration. It drives robust, durable tumor regression, making it a valuable tool for probing PI3Kα‑dependent tumor biology.

References : Buckbinder L. et al.: Cancer Discov., 13(11), 2432-2447, 2023.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.