threo-Ifenprodil hemitartrate

SI-6126

threo-Ifenprodil hemitartrate, >98% (HPLC)

CAS No. : [1312991-83-5]

IUPAC Name : 4-((1R,2R)-2-(4-Benzylpiperidin-1-yl)-1-hydroxypropyl)phenol hemi((2S,3S)-2,3-dihydroxysuccinate)

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : threo‑Ifenprodil hemitartrate exhibits high‑affinity agonism at σ₁ and σ₂ receptors and selectively antagonizes NR2B‑containing NMDA receptors. It also blocks hERG channels at nanomolar potency (IC₅₀ = 88 nM), an activity associated with antiarrhythmic effects.

References : Hashimoto K. et al.: Eur. J. Pharmacol., 273(3), 307-10, 1995; Avenet P. et al.: Eur. J. Pharmacol., 296(2), 209-13, 1996; Monassier L. et al.: J. Pharmacol. Exp. Ther., 322(1), 341-50, 2007.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.