Valemetostat tosylate

SI-6803

Valemetostat tosylate, >98% (HPLC)

CAS No. : [1809336-93-3]

Synonyms : DS-3201 tosylate

IUPAC Name : (R)-7-Chloro-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-((1r,4R)-4-(dimethylamino)cyclohexyl)-2,4-dimethylbenzo[d][1,3]dioxole-5-carboxamide 4-methylbenzenesulfonate

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Valemetostat tosylate potently inhibits both EZH1 and EZH2 with IC₅₀ values below 10 nM, representing a first‑in‑class dual PRC2 inhibitor. It serves as a valuable tool for investigating epigenetic dysregulation and therapeutic vulnerabilities in relapsed or refractory peripheral T‑cell lymphoma.

References : Shimizu J. et al.:. J. Physiol., 600(14), 3331-3353, 2022; Yamagishi M. et al.: Cell Rep., 29(8), 2321-2337, e7, 2019.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.