Velzatinib

SI-7253

Velzatinib, >98% (HPLC)

CAS No. : [2590556-80-0]

Synonyms : M4205; IDRX-42

IUPAC Name : N-(4-(1-Methyl-1H-pyrazol-4-yl)benzyl)-6-(7-(3-(pyrrolidin-1-yl)propoxy)imidazo[1,2-a]pyridin-3-yl)pyrimidin-4-amine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Velzatinib inhibits multiple oncogenic kinases—including PDGFRB, PDGFRA, CSF1R, c‑Kit, FLT3, and LCK—with nanomolar potency (IC₅₀ = 2.6–141 nM). It shows robust antitumor efficacy in xenograft models, highlighting its relevance in multi‑kinase‑driven cancer research.

References : Blum A. et al.: Journal of Medicinal Chemistry, 66(4), 2386-2395, 2023.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.